N-substituted indolyl-3-glyoxylamides, their use as...

Details N-substituted indolyl-3-glyoxylamides, their use as... N-substituted indolyl-3-glyoxylamides, their use as...

2007-05-01

2007-05-01

McKane, Joseph K. (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C546S159000

Reexamination Certificate

active

10892040

ABSTRACT:
The invention relates to novel N-substituted indolyl-3-glyoxylamides of the general formula I, their preparation and use as medicaments, in particular for the treatment of tumors

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Wen-Tai Li et al.,Synthesis and Biological Evaluation of N-Heterocyclic Indolyl Glyoxylamides as Orally Active Anticancer Agents, J. Med. Chem 2003, 46, 1706-1715.

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