N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and

Details N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and

1987-07-13

1990-12-25

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514253, 514321, 514322, 544368, 546198, 546199, 548241, C07D26120, C07D41306, A61K 3142, A61K 31445

Patent

active

049803654

ABSTRACT:
There are disclosed compounds having the formula ##STR1## wherein R.sub.1 is hydrogen or loweralkyl; R.sub.2 is loweralkyl, arylloweralkyl, diarylloweralkyl or --CH.sub.2 CHOHCH.sub.2 OR.sub.5, R.sub.5 being aryl, or alternatively --NR.sub.1 R.sub.2 taken together is ##STR2## R.sub.6 being aryl, arylloweralkyl, diarylloweralkyl, ##STR3## and R.sub.3 and R.sub.4 are each independently methoxy or hydroxy, which compounds are useful as analgesic and hypotensive agents.

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Pigini et al., Eur. J. Med. Chem. 10, p. 29 (1975).
Pigini et al., Eur. J. Med. Chem. 10, p. 33 (1975).
Uno et al., Chem. Pharm. Bull. 24, p. 632 (1976).
Pigini et al. I, Chemical Abstract No. 193144Y, (1975).
Pigini et al. II, Chemical Abstract No. 193145w (1975).
Uno et al. Chemical Abstract No. 39459c (1977).

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