Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2007-08-28
2010-10-19
Wilson, James O (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S275000
Reexamination Certificate
active
07816359
ABSTRACT:
The present invention relates to novel amides and a process for preparing these amides.
REFERENCES:
patent: 2808433 (1957-10-01), Struve
patent: 3505389 (1970-04-01), Weil et al.
patent: 3763234 (1973-10-01), Brill
patent: 4281000 (1981-07-01), Dusza et al.
patent: 4623486 (1986-11-01), Lombardino et al.
patent: 4816485 (1989-03-01), Satzinger et al.
patent: 5137918 (1992-08-01), Weiershausen et al.
patent: 5521184 (1996-05-01), Zimmermann
patent: 2005/0159391 (2005-07-01), Ding et al.
patent: 531480 (1931-07-01), None
patent: 44 28 380 (1996-02-01), None
patent: 0 564 409 (1993-10-01), None
patent: 862127 (1961-03-01), None
patent: 49087761 (1974-08-01), None
patent: 50129738 (1975-04-01), None
patent: 56065804 (1979-11-01), None
patent: 3130252 (1990-06-01), None
patent: 2001510192 (1997-07-01), None
patent: 92 17066 (1992-10-01), None
patent: 99 03854 (1999-01-01), None
patent: WO 99/03854 (1999-01-01), None
patent: WO9959959 (1999-11-01), None
patent: 00 18738 (2000-04-01), None
patent: WO0027820 (2000-05-01), None
patent: 01 27089 (2001-04-01), None
Basha et al., “A mild, general method for conversion of esters to amides,” Tetrahedron Letters, No. 48, pp. 4171-4173 (1977).
Database Crossfire Beilstein, Online, Beilstein Institute zur Foerderung der Chemischen Wissenschaften, Frankfurt am Main, DE (1961), Database accession No. 2775102.
Database Crossfire Beilstein, Online, Beilstein Institute zur Foerderung der Chemischen Wissenschaften, Frankfurt am Main, DE (1970), Database accession No. 3005098.
Database Crossfire Beilstein Online, Beilstein Institut zur Foerderung der Chemischen Wissenschaften, Frankfurt am Main, DE (1957), Database accession No. 3401828.
Database Crossfire Beilstein Online, Beilstein Institut zur Foerderung der Chemischen Wissenschaften, Frankfurt am Main, DE (1931), Database accession No. 3411040.
Lipton, M.F. et al., “Conversion of Esters to Amides with Dimethylaluminum Amides: N,N-Dimethylcyclohexanecarboxamide,” Organic Synthesis, John Wiley 1979, vol. 59, pp. 49-53 (1979).
Gless, R.D., “Lewis Acid Mediated Aminolysis of Esters: Conversion of Methyl (S)-(−)-2-Chloropropionate to (S)-(+)-N,N-Diethyl-2-Chloropropionamide,” vol. 16(6), pp. 633-638 (1986).
Levin et al., “An Alternative Procedure for the Aluminum-Mediated Conversion of Esters to Amides,” Synthetic Communications, vol. 12(13), pp. 989-993 (1982).
Matsumoto et al., “Direct Aminolysis of Nonactivated and Thermally Unstable Esters at High Pressure,” Chem. Ber., vol. 122, pp. 1357-1363 (1989).
Beckwith, A.L.J., “Synthesis of Amides,” University of Adelaide, (1970).
Larock, Richard C., ed., “Comprehensive Organic Transformations—A guide to Functional Group Preparations,” pp. 156-160, pp. 1777-1779, 2388-2392, 5186-5189, 4873-4876 (1989).
Paquette, Leo A., Editor-in-Chief, Encyclopedia of Reagents for Organic Synthesis, vol. 1, A—Bru, The Ohio State University, Columbus, OH (1995).
Ludovici, D W., et al., “Evolution of Anti-HIV Drug Candidates. Part 3: Diarylpyrimidine (DAPY) Analogues”, Bioorganic & Medicinal Chemistry Letters, 11 (2001), pp. 2235-2239.
Moffat et al. “4-pyridin-5-yl, etc.” Bioorganic & Medicinal Chemistry Letters 9 (1999) 3351-3356.
Abel Stephan
Bürger Hans Michael
Kaufmann Daniel
Loiseleur Olivier
Meisenbach Mark
Dohmann George R.
Leeser Erich A
Novartis AG
Wilson James O
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