Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Ester doai
Patent
1986-10-02
1989-05-30
Sutto, Anton H.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Ester doai
558394, A61K 31275, C07C12152
Patent
active
048351806
ABSTRACT:
N-(.omega.-cyanoalkyl)aminophenols of formula ##STR1## useful as lipoxygenase inhibitors and anti-asthmatic agents, are prepared by acylation of an aminophenol with an .omega.-haloalkanoyl chloride followed by reduction of the resulting amide then displacement of the halide by cyanide.
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Johnson Robert E.
Schlegel Donald C.
DuPont Paul E.
Hansen Philip E.
Sterling Drug Inc.
Sutto Anton H.
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