N-(imidazolylalkyl)substituted cyclic amines as histamine-H.sub.

Details N-(imidazolylalkyl)substituted cyclic amines as histamine-H.sub. N-(imidazolylalkyl)substituted cyclic amines as histamine-H.sub.

1998-10-16

2000-10-17

Chang, Ceila

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514212, 514397, 540603, 546210, 5483147, A61K 31445, C07D40106

Patent

active

061332917

ABSTRACT:
The present invention discloses novel N(imidazolylalkyl)-substituted cyclic amine compounds which have excellent histamine-H.sub.3 receptor antagonist activity as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising such cyclic amines as well as methods of using them to treat allergy, inflammatory and CNS-related diseases.

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