Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1989-06-06
1990-04-10
Lee, Mary C.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514255, 514269, 514272, 514274, 544301, 544311, 544312, 544316, 544317, 544319, 544320, 544321, 544322, 544326, 544327, 544328, 544329, 544331, 544332, 544333, 544405, 546193, 546194, A61K 3144, C07D21302, C07D23902
Patent
active
049161423
ABSTRACT:
This invention pertains to novel substituted N-heterocyclic-N-(4-piperidinyl)amides useful as analgesics and antagonists of opiolds, wherein the compounds have the general formula: ##STR1## including optically active isomeric forms, and the pharmaceutically acceptable acid addition salts thereof, wherein:
REFERENCES:
patent: 4157393 (1979-06-01), Sanczuk et al.
patent: 4546105 (1985-10-01), Effland et al.
patent: 4584303 (1986-04-01), Huang et al.
patent: 4792554 (1988-12-01), Elben et al.
Youcheng et al., Structural Modification of 4-N-Propionyl Group, etc. 1983, 7 pgs. (Yaoxue Xuebo 18(8) 591-6).
Studies on Potent Analgesics, Youcheng et al., 3/81, 12 pg. article (Acta Pharmaceutica Sinica), vol. XVI, No. 3.
S. Grossmann et al., Pyridin-Analoga des Fentanyls, 1978, 6 page article (Arch. Pharm. Weinheim).
Janssens et al., New Antihistiminic N-Heterocyclic 4-Piperidiamines, 1985, 5 pgs. (J. Med. Chem), vol. 28, No. 12, pp. 1925-1947.
Bagley Jerome R.
Spencer H. Kenneth
BOC, Inc.
Cassett Larry R.
Lee Mary C.
Richter J.
Swope R. Hain
LandOfFree
N-heterocyclic-N-(4-piperidinyl)amides and pharmaceutical compos does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with N-heterocyclic-N-(4-piperidinyl)amides and pharmaceutical compos, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and N-heterocyclic-N-(4-piperidinyl)amides and pharmaceutical compos will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-2299431