Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1992-04-14
1993-03-23
Daus, Donald G.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514261, 514262, 514263, 514265, 514266, 514316, 514252, 514326, 514321, 514322, 5142342, 5142348, 544266, 544267, 544276, 544277, 544285, 544286, 544287, 544290, 544291, 544292, 544293, 544360, 544211, 544216, 544217, 544116, 544117, 546196, 546198, 546199, 546201, 546202, 546208, 546212, 546213, A61K 31505, A61K 3152, C07D23972
Patent
active
RE0342017
ABSTRACT:
This invention pertains to novel substituted N/aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides useful as analgesics, and methods of administering analgesia, which comprises the systemic administration to mammals of such compounds, and pharmaceutical compositions containing such compounds, wherein the novel compounds have the general formula: ##STR1## including optically active isomeric forms, and the pharmaceutically acceptable acid addition salts thereof, wherein R, R.sub.1, R.sub.2, R.sub.3 and R.sub.4 are defined in the disclosure.
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Bagley Jerome R.
Huang Bao-Shan
Lalinde Nhora L.
Spencer H. Kenneth
Anaquest, Inc.
Cassett Larry R.
Daus Donald G.
Swope R. Hain
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