Muscarinic agonists and antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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Details

514294, 546 94, A01N 4342, A61K 3144, C07D45100, C07D45300

Patent

active

060937246

ABSTRACT:
The present invention provides novel compounds and pharmaceutical compositions thereof useful in the treatment of pain. The compounds of the present invention are azaadamantanes, azanoradamantanes and azahomoadamantanes.

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Bok et al., "Synthesis and Conformational Analysis of Exo-and Endo-7-Substituted-3-Azabicyclo[3.3.1]nonanes," Tetrahedron (1979), 35(2), 267-282.
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