Modulators of cholecystokinin

Details Modulators of cholecystokinin Modulators of cholecystokinin

1994-06-08

1996-04-16

Springer, David B.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548507, 548495, 548253, 548118, C07D20920, C07D40312, A61K 3141, A61K 31405

Patent

active

055084320

ABSTRACT:
CCK modulators, e.g. agonists or antagonists, of the following formula (I): ##STR1## or a base-addtion salt thereof.

REFERENCES:
patent: 4490364 (1984-12-01), Rivier
Horwell, et al. J. Med. Chem. 1991, 34, 404-401 "Rationally Designed `Dipeptoid` Analogues of CCK. .alpha.-Methyltryptophan Derivatives as Highly Selective and Orally Active Gastrin and CCK-B antagonists with Potent Anxiolytic Properties".
Jensen, et al. Biochem. Biophys. Acta. 1983, 757, 250-258 "COOH-Terminal Fragments of Cholecystokinin--A New Class of Cholecystokinin Receptor Antagonists".
Spanarke., et al. J. Bio. Chem. 1983, vol. 258, 11, 6746-6749 "Cholecystokinin-27-32-Amide".
Shiosake, et al. J. Med. Chem. 1990, 33, 2950-2952 "Development of CCK-Tetrapeptide Analogues as Potent and Selective CCK-A Receptor Agonists".
Drysdale, et al. J. Med. Chem. 1992, 35, 2573-2581 "Rationally Designed `Dipeptoid` Analogues of CCK. Acid Mimics of the Potent and Selective Non-Peptide CCK-B Receptor Antagonist Cl-988".

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