Methods of assaying receptor activity and constructs useful in s

Chemistry: molecular biology and microbiology – Measuring or testing process involving enzymes or... – Involving antigen-antibody binding – specific binding protein...

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536 234, 530350, 435 791, 435 691, G01N 3352, C07H 2104, C12N 1512, C07K 1400

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active

058916466

ABSTRACT:
Described are methods of detecting G-protein coupled receptor (GPCR) activity in vivo and in vitro; methods of assaying GPCR activity; and methods of screening for GPCR ligands, G protein-coupled receptor kinase (GRK) activity, and compounds that interact with components of the GPCR regulatory process. Constructs useful in such methods are described.

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