Methods for the formulation and manufacture of artesunic...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C424S600000

Reexamination Certificate

active

07956086

ABSTRACT:
A method for the manufacture of a sterile intravenous or intramuscular formulation of artesunic acid and the formulation are the subject of this invention. First the artesunic acid powder is sterilized with ethylene oxide and placed into a sterile container. The contained sterilized powder is then dissolved in sterile sodium phosphate buffered solution to produce an injectable intravenous or intramuscular formulation. The sodium phosphate dissolves and dilutes the artesunic acid powder without caking or frothing resulting in an improved drug product. The invention also relates to the formulation and a method of treating a patient with either uncomplicated or severe and complicated malaria.

REFERENCES:
patent: 7678828 (2010-03-01), Ellis et al.
patent: 2003/0203875 (2003-10-01), Hartell et al.
Ashley et al., “Malaria” Travel Medicine and Infectious Disease , Elsevier, vol. 4, No. 3-4, May 2006 pp. 159-173.
Hin et al., “Comparative pharmacokinetics of intramuscular artesunate and artemether in patients with severe falciparum malaria”, Antimicrobial Agents And Cemotherapy, vol. 48, No. 11, Nov. 2004, pp. 4234-4239.
Nealon, Claire, et al.: “Intramuscular bioavailability and clinical efficacy of artesunate in gabonese children with severe malaria.” Antimicrobial Agents and Chemotherapy Dec. 2002, vol. 46, No. 12, Dec. 2002, pp. 3933-3939.
Ilett Kenneth et al.: “The pharmacokinetic properties of intramuscular artesunate and rectal dihydroartemisinin in uncomplicated falciparum malaria”, British Journal of Clinical Pharmacology, vol. 53, No. 1, Jan. 2002, pp. 23-30.

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