Methods for synthesis of 3-amino-1-arylpropyl indoles

Details Methods for synthesis of 3-amino-1-arylpropyl indoles Methods for synthesis of 3-amino-1-arylpropyl indoles

2006-11-29

2009-10-06

Saeed, Kamal A (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

active

07598399

ABSTRACT:
A method comprising:hydrogenating an indole propionamide compound of formula hwith vitride, to form an aminopropyl indole compound of formula iwherein m, Ar, R1and R2are as defined herein. The compounds prepared by the method of the invention are useful as monoamine reuptake inhibitors useful for treatment of CNS indications.

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