Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1998-02-12
2000-09-12
Higel, Floyd D.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514248, 530323, 530332, 5482634, A61K 3141, C07K 500, C07K 700, C07K 1600, C07D24912
Patent
active
061178969
ABSTRACT:
.beta.-sheet mimetics and methods relating to the same are disclosed. The .beta.-sheet mimetics have utility as protease and kinase inhibitors, as well as inhibitors of transcription factors and protein-protein binding interactions. Methods of the invention include administration of a .beta.-sheet mimetic, or use of the same for the manufacture of a medicament for treatment of a variety of conditions associated with the targeted protease, kinase, transcription factor and/or protein-protein binding interaction.
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Kahn Michael S.
Mathew Jessymol
McMillan Michael K.
Ogbu Cyprian O.
Qabar Maher N.
Higel Floyd D.
Molecumetics Ltd.
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