Methods for preparing P2X 7 inhibitors

Details Methods for preparing P2X 7 inhibitors Methods for preparing P2X 7 inhibitors

2007-06-26

2007-06-26

Balasubramanian, Venkataraman (Department: 1624)

Organic compounds -- part of the class 532-570 series

Organic compounds

Four or more ring nitrogens in the bicyclo ring system

C514S242000

Reexamination Certificate

active

11167828

ABSTRACT:
The present invention relates to the methods for preparing compounds of the formula I:or the pharmaceutically acceptable salts thereof, wherein R1, R2, R4, R10, and R11have any of the values defined in the specification. The compounds of the present invention are useful in the treatment of diseases, including inflammatory diseases such as rheumatoid arthritis.

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