Method of treating conditions susceptible to modulation of NPY r

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

5142305, 5142358, 514396, 514397, 514398, 514399, 514400, 544 585, 544 62, 544105, 544139, 5483117, 5483365, 5483415, 5483431, 5483435, A61K 3154, A61K 31541, A61K 315415, A61K 315377, A61K 31538, A61K 314166

Patent

active

061212601

ABSTRACT:
Certain diaryl imidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position. Many of the compounds are novel.

REFERENCES:
patent: 3297710 (1967-01-01), Silversmith
patent: 3657441 (1972-04-01), Jensen et al.
patent: 4134983 (1979-01-01), Baldwin
patent: 4665023 (1987-05-01), Deneke et al.
patent: 4757124 (1988-07-01), Koyanagi et al.
patent: 4758639 (1988-07-01), Koynagi et al.
patent: 4853383 (1989-08-01), Baldwin et al.
patent: 5017467 (1991-05-01), Masukawa et al.
patent: 5292669 (1994-03-01), Guder et al.
patent: 5296609 (1994-03-01), McCort et al.
patent: 5498301 (1996-03-01), Hirao et al.
patent: 5620999 (1997-04-01), Weier et al.
Lombardino, Joseph G., et al. "Preparation and Antiinflammatory Activity of Some Nonacidic Trisubstituted Imidazoles." Journal of Medicinal Chemistry, vol. 17, No. 11 (1974, pp. 1182-1188 XP-002080630.
Suzuki, Mamoru et al. "Syntheses of 2-Aryl-4-(3-thienyl)imidazole Derivatives with Antiinflammatory Properties." Chemical and Pharmaceutical Bulletin, vol. 34, No. 8 (1986) pp. 3111-3120 XP-002080631.
Baldwin, J. J., et al. ".beta.-Adrenergic Blocking Agents with Acute Antihypertensive Activity." Journal of Medicinal Chemistry, vol. 22, No. 6 (1979) pp. 687-694 XP002080632.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Method of treating conditions susceptible to modulation of NPY r does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Method of treating conditions susceptible to modulation of NPY r, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Method of treating conditions susceptible to modulation of NPY r will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-1073385

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.