Method of solubilizing itraconazole

Details Method of solubilizing itraconazole Method of solubilizing itraconazole

1997-11-11

2000-08-08

Lovering, Richard D.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514784, 5483501, A61K 31415, A01N 4350

Patent

active

061002852

ABSTRACT:
Solutions comprising itraconazole solubilized in a solvent comprising at least one volatile organic acid are provided. Methods for preparing microspheres containing imidazole derivatives are provided. Also provided is the use of imidazole derivatives containing microspheres for treating fungal infections. Oral dosage forms for oral administration are also provided.

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