Method of solubilizing and encapsulating itraconazole

Drug – bio-affecting and body treating compositions – Preparations characterized by special physical form – Particulate form

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264 41, 264 46, 424435, 514400, 514963, B01J 1304, A61K 964, A61K 31415, A01N 4350

Patent

active

057501475

ABSTRACT:
Methods for preparing microspheres containing imidazole derivatives are provided. Also provided is the use of imidazole derivatives containing microspheres for treating fungal infections. Oral dosage forms for oral administration are also provided.

REFERENCES:
patent: Re24899 (1960-11-01), Green
patent: 2671451 (1954-03-01), Bolger
patent: 2862918 (1958-12-01), Meyer et al.
patent: 2868740 (1959-01-01), Luce
patent: 2971916 (1961-02-01), Schleicher et al.
patent: 3016308 (1962-01-01), Macaulay
patent: 3052655 (1962-09-01), Fox et al.
patent: 3057344 (1962-10-01), Abella et al.
patent: 3076790 (1963-02-01), Fox et al.
patent: 3170802 (1965-02-01), Fukushima
patent: 3190837 (1965-06-01), Brynko et al.
patent: 3474777 (1969-10-01), Figge et al.
patent: 3491093 (1970-01-01), Pachter et al.
patent: 3565559 (1971-02-01), Sato et al.
patent: 3567650 (1971-03-01), Bakan
patent: 3574832 (1971-04-01), Engel et al.
patent: 3576758 (1971-04-01), Emrick
patent: 3687926 (1972-08-01), Arima et al.
patent: 3725113 (1973-04-01), Chang
patent: 3794561 (1974-02-01), Matsukawa et al.
patent: 3795739 (1974-03-01), Birkmayer et al.
patent: 3822348 (1974-07-01), Higashi et al.
patent: 3849550 (1974-11-01), Teitelbaum
patent: 3937668 (1976-02-01), Zolle
patent: 3939253 (1976-02-01), Bodor et al.
patent: 3956172 (1976-05-01), Saeki et al.
patent: 3962416 (1976-06-01), Katzen
patent: 4035507 (1977-07-01), Bodor et al.
patent: 4048268 (1977-09-01), Ludwig
patent: 4061466 (1977-12-01), Sjoholm et al.
patent: 4117801 (1978-10-01), Dannelly et al.
patent: 4147767 (1979-04-01), Yapel
patent: 4183849 (1980-01-01), Hansen et al.
patent: 4199561 (1980-04-01), Roth et al.
patent: 4217370 (1980-08-01), Rawlings et al.
patent: 4272506 (1981-06-01), Schwarzberg
patent: 4345588 (1982-08-01), Widder et al.
patent: 4348384 (1982-09-01), Horikoshi et al.
patent: 4351337 (1982-09-01), Sidman
patent: 4352993 (1982-10-01), Lim
patent: 4357259 (1982-11-01), Senyei et al.
patent: 4388304 (1983-06-01), Nyeki et al.
patent: 4402856 (1983-09-01), Schnoring et al.
patent: 4405598 (1983-09-01), Brown
patent: 4442090 (1984-04-01), Kakeya et al.
patent: 4446138 (1984-05-01), Pack
patent: 4450150 (1984-05-01), Sidman
patent: 4457907 (1984-07-01), Porter
patent: 4460563 (1984-07-01), Calanchi
patent: 4462839 (1984-07-01), McGinley et al.
patent: 4462991 (1984-07-01), Higuchi et al.
patent: 4473620 (1984-09-01), Wu et al.
patent: 4483807 (1984-11-01), Asano et al.
patent: 4492684 (1985-01-01), Goosen et al.
patent: 4518433 (1985-05-01), McGinley et al.
patent: 4590265 (1986-05-01), Bogan et al.
patent: 4608278 (1986-08-01), Frank et al.
patent: 4613500 (1986-09-01), Suzuki et al.
patent: 4647455 (1987-03-01), De Bold
patent: 4666641 (1987-05-01), Fickat et al.
patent: 4671954 (1987-06-01), Goldberg
patent: 4673566 (1987-06-01), Goosen et al.
patent: 4683092 (1987-07-01), Tsang
patent: 4703042 (1987-10-01), Bodor
patent: 4708952 (1987-11-01), Salatinjants
patent: 4745161 (1988-05-01), Saudek et al.
patent: 4753804 (1988-06-01), Iaccheri et al.
patent: 4757007 (1988-07-01), Satoh
patent: 4757024 (1988-07-01), Roper
patent: 4766012 (1988-08-01), Valenti
patent: 4774320 (1988-09-01), Tagliabue et al.
patent: 4789734 (1988-12-01), Pierschbacher
patent: 4835312 (1989-05-01), Itoh et al.
patent: 4844904 (1989-07-01), Hamaguchi et al.
patent: 4873087 (1989-10-01), Morishita et al.
patent: 4886663 (1989-12-01), Houghten
patent: 4895725 (1990-01-01), Kantor et al.
patent: 4897444 (1990-01-01), Brynes et al.
patent: 4900730 (1990-02-01), Miyauchi
patent: 4925673 (1990-05-01), Steiner
patent: 4963364 (1990-10-01), Fox et al.
patent: 4976968 (1990-12-01), Steiner
patent: 4983402 (1991-01-01), Steiner
patent: 4996292 (1991-02-01), Fox et al.
patent: 5039481 (1991-08-01), Pacifici et al.
patent: 5055300 (1991-10-01), Gupta
patent: 5066487 (1991-11-01), Morelle et al.
patent: 5069936 (1991-12-01), Yen
patent: 5077278 (1991-12-01), Hafner et al.
patent: 5100669 (1992-03-01), Hyon et al.
patent: 5186947 (1993-02-01), Goettsche et al.
patent: 5204099 (1993-04-01), Barbier et al.
patent: 5206384 (1993-04-01), Shibahara et al.
patent: 5250236 (1993-10-01), Gasco
patent: 5271961 (1993-12-01), Mathiowitz et al.
patent: 5328992 (1994-07-01), Peter et al.
patent: 5384133 (1995-01-01), Boyes et al.
patent: 5418010 (1995-05-01), Janda et al.
patent: 5474997 (1995-12-01), Gray et al.
patent: 5536813 (1996-07-01), Charpenel et al.
Chemical Abstracts, 76(14):72994u, (1971).
Chemical Abstracts, 84(7):44660d, (1975).
Chemical Abstracts, 86(16):107529g, (1976).
Chemical Abstracts, 112(15):134663h, (1989).
Chemical Abstracts, 114(22):214519x, (1990).
J. Gyore et al., Thermal Analysis, vol. 2 -Proceeding Fourth ICTA Budapest 1974, pp. 387-394.
Chemical Abstracts, 99(19) 158832b, (1982).
Derwent Abstracts, JP 67008622, (1967).
Airaudo, C.B. et al. (1987) Journal of Food Science, vol. 52(6), pp. 1750-1752.
Andini, S. et al. (1975) Origins of Life, vol. 6, pp. 147-153.
Brooke, S. 1 et al. (1977) BioSystems, vol. 9, pp. 1-22.
Chen et al. (1975) "Evidence for Hemiacetal Formation", Biochemistry, vol. 18, No. 5, pp. 921-925.
Davis et al. (1983) "Leucinal Inhibits . . . ", Pharmacology Biochemistry Behavior, vol. 19, pp. 791-794.
Dose, K. (1974) Origins of Life, vol. 5, pp. 239-252.
Fasman et al. (1964) Biochemistry, vol. 3, No. 11, pp. 1665-1674.
Fox, S.W. et al. (1976) BioSystems, vol. 8, pp. 40-44.
Fox, S.W. et al., Molecular Evolution and the Origin of Life, Maxel Decker, New York (1977).
Fox, S.W. et al. (1968) Biochim. Biophys. Acta, vol. 160, pp. 246-249.
Fox, S.W. (1976) Origins of Life, vol. 7, pp. 49-68.
Fox, S.W. (1980) Naturwissenschaften, vol. 67, pp. 378-383.
Fox, S.W. et al. (1960) Archives of Biochemistry and Biophysics, vol. 86, pp. 281-285.
Fox, S.W. et al. (1974) Origins of Life, vol. 5, pp. 227-237.
Fox, S.W. (1984) Origins of Life, vol. 14, pp. 485-488.
Gol'dovskii, A.M. (1978) Zhurnal Evolyutsionnoi Biokhimii i Fiziologii, vol. 14(6), pp. 437-439.
Gurrieri, S. et al. (1973) Thermochimica Acta, vol. 7, pp. 231-239.
Harada, K. et al. (1979) BioSystems, vol. 11, pp. 47-53.
Harada, K. et al., (1960) Archives of Biochemistry and Biophysics, vol. 86, pp. 274-280.
Hare (1970) Etude Cenetique De La Polycondensation Thermique D'.chi.-Amino Acides, vol. 45, pp. 330-339.
Heinrich, M.R. et al. (1969) Archives of Biochemistry and Biophysics, vol. 130, pp. 441-448.
Heinz, B. et al. (1981) BioSystems, vol. 14, pp. 33-40.
Hennon, G. et al. (1975) Biochimie, vol. 57, pp. 1395-1396.
Hsu, L.L. et al. (1976) BioSystems, vol. 8, pp. 89-101.
Hsu, L.L. et al. (1971) Currents in Modern Biology, vol. 4, pp. 12-25.
Ishima, Y. et al. (1981), BioSystems, vol. 14, pp. 243-251.
Jackson et al. (1991) "Pharmacological . . . ", J. Pharm. & Exp. Thera., vol. 261, No. 1, pp. 546-552.
Jungck, J.R. et al. (1973) Naturwissenschaften, vol. 60, pp. 425-427.
Kokufuta, E. et al., (1984) BioSystems, vol. 16, pp. 175-181.
Krampitz, G. et al. (1967) Naturwissenschaften, pp. 516-517.
Krampitz, G. et al. (1968) Naturwissenschaften, pp. 345-346.
Krampitz, G. et al. (1966) Naturwissenschaften, pp. 7 and 8.
Lacey, Jr., J.C. et al. (1979) BioSystems, vol. 11, pp. 9-17.
Lacey, Jr., J.C. et al. (1979) BioSystems, vol. 11, pp. 1-7.
Martinez Luque-Romero, M. et al. (1986) BioSystemsvol. 19, pp. 267-272.
Masinovsky, Z. et al. (1989) BioSystems, vol. 22, pp. 305-310.
Matsuno, K. (1982) BioSystems, vol. 15, pp. 1-11.
Matsuno, K. (1984) BioSystems, vol. 17, pp. 11-14.
Matsuno, K. (1981) BioSystems, vol. 14, pp. 163-170.
McAlhaney, W.W. et al. (1976) BioSystems, vol. 8, pp. 45-50.
Melius, P. et al. (1987) BioSystems, vol. 20, pp. 213-217.
Melius, P. et al. (1975) Bioorganic Chemistry, vol. 4, pp. 385-391.
Melius, P. (1979) BioSystems, vol. 11, pp. 125-132.
Miquel, J. et al. (1971) Currents in Modern Biology, vol. 3, pp. 299-306.
Nakashima, T. et al. (1980) J. Mol. Evol., vol. 15, pp. 161-168.
Nakashima, T. et al. (1981) BioSystems, vol. 14, pp. 151-161.
Novak, V.J.A. (1984) Origins of Life, vol 14, pp. 513-522.
Olafsson, P.G. et al. (1971) Polymer Letters, vol. 9, pp. 521-528.
Phillips, R.D. et al. (1974) Int.

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