Method of preparing retroviral protease inhibitor intermediates

Details Method of preparing retroviral protease inhibitor intermediates Method of preparing retroviral protease inhibitor intermediates

1995-01-20

1998-11-03

Gerstl, Robert

Organic compounds -- part of the class 532-570 series

Organic compounds

Sulfonic acids or salts thereof

567114, 567585, 567597, 567607, 564192, 564281, 564285, 564305, 564306, C07C30901

Patent

active

058311173

ABSTRACT:
Chiral hydroxyethylamine, hydroxyethylurea or hydroxyethylsulfonamide isostere containing retroviral protease and renin inhibitors can be prepared by multi-step syntheses that utilize key chiral amine intermediates. This invention is a cost effective method of obtaining such key chiral amine intermediates enantiomerically, diastereomerically and chemically pure. The method is suitable for large scale (multikilogram) productions. This invention also encompasses organic acid and inorganic acid salts of the amine intermediates.

REFERENCES:
patent: 4826815 (1989-05-01), Luly et al.

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