Method of preparation of 21-amino epothilone derivatives

Details Method of preparation of 21-amino epothilone derivatives Method of preparation of 21-amino epothilone derivatives

2005-08-16

2005-08-16

Shameem, Golam M M (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C548S146000, C548S203000

Reexamination Certificate

active

06930187

ABSTRACT:
An improved method of synthesis of 21-amino epothilone derivatives which provides a one-pot conversion of 21-hydroxy epothilones to highly desirable 21-amino epothilones in high yield.

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