Method of inhibiting amyloid protein aggregation and imaging...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C514S535000, C514S564000, C514S567000, C514S657000, C548S253000, C548S254000, C560S043000, C562S454000, C562S457000, C564S428000

Reexamination Certificate

active

06949575

ABSTRACT:
The present invention provides compounds of Formula (I) and a method of treating Alzheimer's disease using a compound of Formula (I), wherein: R1and R2include alkyl and phenylalkyl; R3is hydrogen or alkyl; and R4and R5include alkyl, alkoxy, carboxyl, alkoxycarbonyl, and nitro. Also provided is a method of inhibiting the aggregation of amyloid proteins using a compound of Formula (I)and a method of imaging amyloid deposits using compounds of Formula (I).

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