Method of blocking peripheral norepinephrine release

Details Method of blocking peripheral norepinephrine release Method of blocking peripheral norepinephrine release

1982-11-03

1984-08-28

Fan, Jane T.

Drug, bio-affecting and body treating compositions

Antigen, epitope, or other immunospecific immunoeffector

Bacterium or component thereof or substance produced by said...

546 82, A61K 3147, C07D47104

Patent

active

044684010

ABSTRACT:
Trans-4aR-5-n-propyl-4,4a,5,6,7,8,8a,9-octahydro-1H(and 2H)pyrazolo[3,4-g]quinoline and pharamceutically-acceptable salts thereof, blocks norepinephrine release from peripheral sympathetic nerve terminals that innervate arterial muscle fibers in hypertensive mammals to reduce blood pressure.

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