Method for producing an injectable medicament preparation

Drug – bio-affecting and body treating compositions – Radionuclide or intended radionuclide containing; adjuvant...

Reexamination Certificate

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C530S350000, C514S002600

Reexamination Certificate

active

07387771

ABSTRACT:
The invention relates to a method for producing injectable medicament preparations containing a therapeutically and/or diagnostically effective substance which is comprised of an active agent, of a spacer molecule and of at least one protein-binding molecule. After being brought into contact with the body, said therapeutically and/or diagnostically effective substance covalently bonds to the body fluid constituents or tissue constituents via the protein-binding molecules, thus providing a form of transport of the active agent that can be hydrolytically or enzymatically cleaved, according to pH, in the body while releasing the active agent.

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