Method for producing 4-nitroimidazole compound

Details Method for producing 4-nitroimidazole compound Method for producing 4-nitroimidazole compound

2005-02-15

2009-08-04

Shiao, Rei-Tsang (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C514S398000

Reexamination Certificate

active

07569702

ABSTRACT:
The present invention provides a method for producing a 4-nitroimidazole compound represented by general formula (1) at high yield and at high purity by a safe method causing few dangers such as explosion. The production method of the present invention comprises iodinating a 4-nitroimidazole compound represented by general formula (2): wherein each of X1and X2represents a chlorine atom or bromine atom, and then reducing the obtained 5-iodo-4-nitroimidazole compound represented by general formula (3): wherein X2is the same as defined above.

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