Method for increasing HDL cholesterol levels using heteroaromati

Details Method for increasing HDL cholesterol levels using heteroaromati Method for increasing HDL cholesterol levels using heteroaromati

1998-09-09

2000-08-15

Higel, Floyd D.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514399, 514400, 514427, 546343, 546378, 5483401, 5483461, A61P 300, A61P 910, A61K 31435, A61K 314164, A61R 3140

Patent

active

061037338

ABSTRACT:
An HDL cholesterol level inducing compound and a method of administering the compound having the structural formula I. ##STR1## wherein n is 1 or 2;
R.sub.1 is a heteroaromatic substituent independently selected from a five-membered heteroaromatic ring having at least one N heteroatom, a six-membered heteroaromatic ring having at least one N heteroatom, or a fused ring system having at least one five-membered heteroaromatic ring having at least one N heteroatom;
R.sub.2 is independently selected from --H or phenyl; and
R.sub.3 is independently selected from --H, --CH.sub.3, --OH, phenyl, phenyl substituted with Cl, OCH.sub.3, CH.sub.3, or F, fused phenyl ring system, or six-membered heteroaromatic ring having at least one N heteroatom.

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