Method for expedient synthesis of [18F]-labeled...

Organic compounds -- part of the class 532-570 series – Organic compounds – Oxygen containing

Reexamination Certificate

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C568S325000, C376S168000, C382S130000, C382S131000

Reexamination Certificate

active

06872855

ABSTRACT:
The present invention is directed to a convenient method of synthesizing radiolabeled α-trifluoromethyl ketones by a fluorination reaction. The present invention also relates to imaging agents and markers for identifying cell proliferation, or viral infection. The markers and imaging agents including the radiolabeled α-trifluoromethyl ketones that are prepared by the present method.

REFERENCES:
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G.K. Surya Prakash et al.; “A general method of halogenation for synthesis of αhalodifluoromethyl ketones and [18]-labeled trifluoromethyl ketones”; Journal of Fluorine Chemistry 121 (2003) 239-243.
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