Melphalan derivatives and their use as cancer...

Details Melphalan derivatives and their use as cancer... Melphalan derivatives and their use as cancer...

2006-01-31

2006-01-31

Barts, Samuel (Department: 1621)

Organic compounds -- part of the class 532-570 series

Organic compounds

Carboxylic acid esters

C562S450000, C564S123000, C564S149000, C564S152000, C564S155000, C564S157000, C514S002600

Reexamination Certificate

active

06992207

ABSTRACT:
The invention refers to new alkylating di- and tripeptides based on a melphalan unit, and one or two additional amino acids or amino acid derivatives, which can be used in the treatment of carcinogenic diseases. Further, the invention refers to a pharmaceutical composition comprising the alkylating peptides of the invention.

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