Melanocortin receptor-specific compounds

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S252130, C514S254090, C544S358000, C544S372000, C544S373000

Reexamination Certificate

active

07964601

ABSTRACT:
A melanocortin receptor-specific compound of the general formula of structure I:where X, R1, R2a, R2b, R3, R4a, R4b, R5aand R5bare as defined in the specification, which compound binds with high affinity to one or more melanocortin receptors and is optionally an agonist, an antagonist, an inverse agonist or an antagonist of an inverse agonist, and may be employed for treatment of one or melanocortin receptor-associated conditions or disorders, and methods for the use of the compounds of the invention.

REFERENCES:
patent: 4148923 (1979-04-01), Giudicelli et al.
patent: 4239763 (1980-12-01), Milavec et al.
patent: 4626549 (1986-12-01), Molloy et al.
patent: 4680289 (1987-07-01), Applezweig
patent: 4711957 (1987-12-01), Lai
patent: 4766125 (1988-08-01), Van Daele
patent: 4937267 (1990-06-01), Holloway et al.
patent: 4938763 (1990-07-01), Dunn et al.
patent: 4943578 (1990-07-01), Naylor et al.
patent: 4968684 (1990-11-01), Van Daele et al.
patent: 4997836 (1991-03-01), Sugihara et al.
patent: 5120713 (1992-06-01), Mugica
patent: 5292726 (1994-03-01), Ashton et al.
patent: 5331573 (1994-07-01), Balaji et al.
patent: 5334830 (1994-08-01), Fukuyama et al.
patent: 5348955 (1994-09-01), Greenlee et al.
patent: 5464788 (1995-11-01), Bock et al.
patent: 5494919 (1996-02-01), Morriello et al.
patent: 5550131 (1996-08-01), Sugihara et al.
patent: 5574031 (1996-11-01), Abramo et al.
patent: 5579250 (1996-11-01), Balaji et al.
patent: 5599809 (1997-02-01), Hickey et al.
patent: 5639778 (1997-06-01), Andersson et al.
patent: 5672602 (1997-09-01), Burkholder et al.
patent: 5721250 (1998-02-01), Morriello et al.
patent: 5721251 (1998-02-01), Chen et al.
patent: 5736539 (1998-04-01), Graham et al.
patent: 5753445 (1998-05-01), Fillit et al.
patent: 5753653 (1998-05-01), Bender et al.
patent: 5763445 (1998-06-01), Kruse et al.
patent: 5798359 (1998-08-01), Shue et al.
patent: 5804578 (1998-09-01), Chakravarty et al.
patent: 5856326 (1999-01-01), Anthony et al.
patent: 5872262 (1999-02-01), Dolle et al.
patent: 5877182 (1999-03-01), Nargund et al.
patent: 5880125 (1999-03-01), Nargund
patent: 5880128 (1999-03-01), Doll et al.
patent: 5891418 (1999-04-01), Sharma
patent: 5892038 (1999-04-01), Dolle et al.
patent: 5936089 (1999-08-01), Carpino et al.
patent: 5965565 (1999-10-01), Chen et al.
patent: 5968938 (1999-10-01), Williams et al.
patent: 6020334 (2000-02-01), Fukushi et al.
patent: 6027711 (2000-02-01), Sharma
patent: 6033656 (2000-03-01), Mikami et al.
patent: 6127381 (2000-10-01), Basu et al.
patent: 6127424 (2000-10-01), Martin et al.
patent: 6140354 (2000-10-01), Dax et al.
patent: 6162805 (2000-12-01), Hefti
patent: 6191117 (2001-02-01), Kozachuk
patent: 6207665 (2001-03-01), Bauman et al.
patent: 6207699 (2001-03-01), Rothman
patent: 6214831 (2001-04-01), Yokoo et al.
patent: 6245764 (2001-06-01), Kahn et al.
patent: 6284735 (2001-09-01), Girten et al.
patent: 6294539 (2001-09-01), Lou et al.
patent: 6303611 (2001-10-01), Zhang et al.
patent: 6316470 (2001-11-01), Kover et al.
patent: 6331285 (2001-12-01), Sharma
patent: 6340868 (2002-01-01), Lys et al.
patent: 6350760 (2002-02-01), Bakshi et al.
patent: 6372747 (2002-04-01), Taveras et al.
patent: 6376509 (2002-04-01), Bakshi et al.
patent: 6410548 (2002-06-01), Nargund et al.
patent: 6432438 (2002-08-01), Shukla
patent: 6432959 (2002-08-01), Cooper et al.
patent: 6451783 (2002-09-01), Hadcock et al.
patent: 6458789 (2002-10-01), Forood et al.
patent: 6458790 (2002-10-01), Palucki et al.
patent: 6469006 (2002-10-01), Blair et al.
patent: 6472398 (2002-10-01), Palucki et al.
patent: 6486165 (2002-11-01), Zhang et al.
patent: 6515122 (2003-02-01), Lang et al.
patent: 6531476 (2003-03-01), Heymans et al.
patent: 6534503 (2003-03-01), Dines et al.
patent: 6534509 (2003-03-01), Bauman et al.
patent: 6555537 (2003-04-01), Bauman et al.
patent: 6569861 (2003-05-01), Bakthavatchalam et al.
patent: 6579968 (2003-06-01), Blood et al.
patent: 6612805 (2003-09-01), Rietsch
patent: 6648848 (2003-11-01), Keldmann et al.
patent: 6673767 (2004-01-01), Brodbeck et al.
patent: 6699873 (2004-03-01), Maguire et al.
patent: 6715485 (2004-04-01), Djupesland
patent: 6734175 (2004-05-01), Hadcock et al.
patent: 6811543 (2004-11-01), Keldmann et al.
patent: 6949552 (2005-09-01), Nakazato et al.
patent: 7326707 (2008-02-01), Sharma et al.
patent: 7354923 (2008-04-01), Sharma et al.
patent: 7456184 (2008-11-01), Sharma et al.
patent: 7709484 (2010-05-01), Sharma et al.
patent: 2001/0018075 (2001-08-01), Shigeyuki et al.
patent: 2001/0047001 (2001-11-01), Varkhedkar et al.
patent: 2002/0004512 (2002-01-01), Bakshi et al.
patent: 2002/0010182 (2002-01-01), Masaaki et al.
patent: 2002/0019523 (2002-02-01), Palucki et al.
patent: 2002/0022620 (2002-02-01), Kahn et al.
patent: 2002/0032238 (2002-03-01), Priepke et al.
patent: 2002/0037837 (2002-03-01), Takada et al.
patent: 2002/0042399 (2002-04-01), Kruse et al.
patent: 2002/0052383 (2002-05-01), Bakthavatchalam et al.
patent: 2002/0065277 (2002-05-01), Hadcock et al.
patent: 2002/0065416 (2002-05-01), Stasiak et al.
patent: 2002/0072604 (2002-06-01), Carpino et al.
patent: 2002/0082263 (2002-06-01), Lou et al.
patent: 2002/0107253 (2002-08-01), Koh et al.
patent: 2002/0107255 (2002-08-01), Blumberg et al.
patent: 2002/0128247 (2002-09-01), Dow et al.
patent: 2002/0128270 (2002-09-01), Neya et al.
patent: 2002/0137664 (2002-09-01), Bakshi et al.
patent: 2002/0143141 (2002-10-01), Chen et al.
patent: 2002/0173512 (2002-11-01), Moltzen et al.
patent: 2002/0177598 (2002-11-01), Bauman et al.
patent: 2002/0183316 (2002-12-01), Pan et al.
patent: 2003/0004162 (2003-01-01), Treadway
patent: 2003/0013721 (2003-01-01), Meghani et al.
patent: 2003/0040520 (2003-02-01), Guzi et al.
patent: 2003/0055008 (2003-03-01), Marcotte
patent: 2003/0055009 (2003-03-01), Steiner et al.
patent: 2003/0055247 (2003-03-01), Cosford et al.
patent: 2003/0055265 (2003-03-01), Binggeli et al.
patent: 2003/0060473 (2003-03-01), Neya et al.
patent: 2003/0064921 (2003-04-01), Millhauser et al.
patent: 2003/0069169 (2003-04-01), Macor et al.
patent: 2003/0083228 (2003-05-01), Carpino et al.
patent: 2003/0083335 (2003-05-01), Hayward
patent: 2003/0092732 (2003-05-01), Yu et al.
patent: 2003/0096827 (2003-05-01), Yu et al.
patent: 2003/0105106 (2003-06-01), Chiang et al.
patent: 2003/0109556 (2003-06-01), Mazur et al.
patent: 2003/0125334 (2003-07-01), Chiang et al.
patent: 2003/0139425 (2003-07-01), Bauman et al.
patent: 2003/0144277 (2003-07-01), DeLucca
patent: 2003/0149019 (2003-08-01), Bremberg et al.
patent: 2003/0158205 (2003-08-01), Bauman et al.
patent: 2003/0158209 (2003-08-01), Dyck et al.
patent: 2003/0162819 (2003-08-01), Eisinger et al.
patent: 2003/0166637 (2003-09-01), Lehmann-Lintz et al.
patent: 2003/0176425 (2003-09-01), Eisinger et al.
patent: 2003/0181441 (2003-09-01), McClure et al.
patent: 2003/0191136 (2003-10-01), Bakthavatchalam et al.
patent: 2003/0195212 (2003-10-01), Lundstedt et al.
patent: 2004/0006067 (2004-01-01), Fotsch et al.
patent: 2004/0024211 (2004-02-01), Boyce et al.
patent: 2004/0034034 (2004-02-01), Blumberg et al.
patent: 2004/0053933 (2004-03-01), Pontillo et al.
patent: 2004/0147567 (2004-07-01), Nakazato et al.
patent: 2004/0152534 (2004-08-01), Chapman et al.
patent: 2004/0157264 (2004-08-01), Sharma et al.
patent: 2004/0171520 (2004-09-01), Sharma et al.
patent: 2004/0204398 (2004-10-01), Bakshi et al.
patent: 2004/0224957 (2004-11-01), Sharma et al.
patent: 2004/0254198 (2004-12-01), Reynolds et al.
patent: 2005/0124636 (2005-06-01), Sharma et al.
patent: 2005/0130988 (2005-06-01), Sharma et al.
patent: 2005/0176728 (2005-08-01), Sharma et al.
patent: 2006/0009456 (2006-01-01), Hutchinson et al.
patent: 2006/0084657 (2006-04-01), Nakazato et al.
patent: 2006/0287330 (2006-12-01), Sharma et al.
patent: 2006/0287331 (2006-12-01), Sharma et al.
patent: 2006/0287332 (2006-12-01), Sharma et al.
patent: 2008/0070921 (2008-03-01), Burris et al.
patent: 2009/0076029 (2009-03-01), Sharma et al.
patent: WO 96/38471 (1996-12-01), None
patent: WO 97/46553 (1997-12-01), None
patent: WO 98/10653 (1998-03-01), None

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