Lupane triterpenoid derivatives

Details Lupane triterpenoid derivatives Lupane triterpenoid derivatives

1993-08-09

1997-07-01

Hollinden, Gary E.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

514 25, 514 53, 514 61, 514169, 514172, 514176, 514178, 536 41, 536 5, 536 187, 5361231, 53612313, A61K 31705, C07J 1700

Patent

active

056438842

ABSTRACT:
This invention relates generally to the field of medicinal chemistry, and more specifically to derivatives of a subclass of triterpenoid acids that have multi-medicament properties, that is derivatives of the lupane, betulinic acid, formulations containing such, and their use to prevent or treat certain diseases, and preferably to derivatives or analogues of betulinic acid, that have the following structural formula (1): ##STR1## wherein: Y is OR.sup.1, NR.sup.1.sub.2, O.sup.- M.sup.1 ;

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