Linear chain substituted monocyclic and bicyclic derivatives...

Details Linear chain substituted monocyclic and bicyclic derivatives... Linear chain substituted monocyclic and bicyclic derivatives...

2006-11-14

2006-11-14

McKane, Joseph K. (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C514S253040, C514S303000, C544S117000, C544S362000, C546S120000

Reexamination Certificate

active

07135469

ABSTRACT:
The present application describes linear chain substituted monocyclic and bicyclic compounds and derivatives thereof of Formula I:in-line-formulae description="In-line Formulae" end="lead"?P4-P-M-M4Iin-line-formulae description="In-line Formulae" end="tail"?or pharmaceutically acceptable salt forms thereof, P-M are rings substituted by a linear group. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.

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