Kappa agonist compounds pharmaceutical formulations and method o

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

514 85, 544337, 544358, 544359, 544360, 544372, 544383, 544386, 544387, 544389, A61K 31495, C07D24104

Patent

active

060573236

ABSTRACT:
Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics and anti-pruritic agents are provided.
The compound of formula I, having the structure: ##STR1## wherein R.sub.1, R.sub.2 ;

REFERENCES:
patent: 4065573 (1977-12-01), Lednicer
patent: 4098904 (1978-07-01), Szmuszkovicz
patent: 4145435 (1979-03-01), Szmuszkovicz
patent: 4212878 (1980-07-01), Lednicer et al.
patent: 4359476 (1982-11-01), Kaplan et al.
patent: 4438130 (1984-03-01), Kaplan
patent: 4663343 (1987-05-01), Horwell et al.
patent: 4855316 (1989-08-01), Horwell et al.
patent: 4906655 (1990-03-01), Horwell et al.
patent: 5646151 (1997-07-01), Kruse et al.
patent: 5688955 (1997-11-01), Kruse et al.
patent: 5744458 (1998-04-01), Kruse et al.
McMahon et al., TINS, vol. 15, No. 12 (1992).
Bernstein et al., Journal of Investigative Dermatology, 78: 82-83 (1982).
Ballantyne et al., Pain, 33: 149-160 (1988).
J. D. Bernhard, J. Am. Acad. Derm. 24: 309 (1991).
IASP Newsletter, Sep./Oct. 1996.
Thomas et al., Brain Research, 695:267-270 (1995).

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Kappa agonist compounds pharmaceutical formulations and method o does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Kappa agonist compounds pharmaceutical formulations and method o, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Kappa agonist compounds pharmaceutical formulations and method o will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-1594041

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.