Kappa agonist compounds pharmaceutical formulations and method o

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Phosphorus containing other than solely as part of an...

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514 89, 514 90, 5142312, 5142395, 514319, 514424, 514429, 514443, 514469, 514613, 514617, 514618, 514619, A61K 31675, A61K 3140

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060544457

ABSTRACT:
Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics and anti-pruritic agents are provided. The compound of formulae IIA, having the structure: ##STR1## wherein R.sub.1, R.sub.2 ;

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