Kappa agonist compounds and pharmaceutical formulations thereof

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

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548413, 548465, 548517, 548527, 548556, 548568, 544106, 544111, 544168, 564182, C07D40110

Patent

active

056889550

ABSTRACT:
Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics are provided.
The compounds of formulae I, II, III and IV have the structure: ##STR1## wherein X, X.sub.4, X.sub.5, X.sub.7, X.sub.9 ;

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Raynor et al., Molecular Pharmacol., 45: 330-334 (1994).
Wheeler-Aceto et al., Psychopharmacology, 104: 35-44 (1991).

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