Isoxazoline derivative and novel process for its preparation

Details Isoxazoline derivative and novel process for its preparation Isoxazoline derivative and novel process for its preparation

2006-02-21

2011-10-25

Qazi, Sabiha (Department: 1628)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C546S139000, C548S240000, C549S430000

Reexamination Certificate

active

08044080

ABSTRACT:
The present invention relates to an isoxazoline derivative having the cyclic carboxylic acid hemiketal moiety of formula (1) for use as caspase inhibitor, a process for preparing it, and a pharmaceutical composition comprising it.

REFERENCES:
patent: 1999-79267 (1999-11-01), None
patent: WO-01/21599 (2001-03-01), None
patent: WO-01/21600 (2001-03-01), None
patent: WO-2005/021516 (2005-03-01), None
Lewis Acid Coordinated Nitrile Oxide and Nitrile Imine 1,3-Dipoles. syn-Selective Cycloadditions to 2-(1-Hydroxyalkyl)acrylates, Bull. Chem. Soc. Jpn., vol. 66, pp. 2685-2693.
Synthesis of a Peptidyl Difluoro Ketone Bearing the Aspartic Acid Side Chain: An Inhibitor of Interleukin-1beta Convering Enzyme, J. Org. Chem., vol. 57, pp. 7309-7314.

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