Isolation and structural elucidation of halistatin 3

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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549264, A61K 31335, C07D31500

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active

055190502

ABSTRACT:
The Micronesian marine sponge Phakellia sp. has been found to contain cern key members of the antineoplastic halichondrin/halistatin family. These compounds include halichondrin B, homohalichondrin B, halistatin 1, and halistatin 3.
Halistatin 3 is a newly discovered member of this family. It inhibited both the P388 leukemia cell line and selected brain, lung, colon, ovarian, renal, and melanoma type cancer cell lines with ED.sub.50 /GI.sub.50 concentrations on the order of 3.times.10.sup.-5 .mu.g/ml.

REFERENCES:
patent: 5328929 (1994-07-01), Pettit et al.
patent: 5352804 (1994-10-01), Pettit et al.

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