Intermediaties for aminooxypyrrolidinylthiocarbapenem compounds

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

548550, 548541, C07D20700

Patent

active

055234151

ABSTRACT:
An antibacterial aminooxypyrrolidinylthiocarbapenem I, its production from the corresponding carbapenem V and thiol VI, its pharmaceutical formulation, and its use for combating bacteria are presented. ##STR1## (wherein R is optionally substituted amino; R.sup.1 is hydrogen or 1C to 5C alkyl; R.sup.2 is hydrogen or a conventional hydroxy protective group; R.sup.3 is hydrogen or an imino protective group or imino substituent; R.sup.4 is 1C to 5C alkylene; and R.sup.5 is hydrogen or a conventional carboxy protective group; X is a leaving group; R.sup.6 is hydrogen or a thiol protective group; and wavy lines each shows a bond in R or S configuration).

REFERENCES:
patent: 4251541 (1981-02-01), Walsh et al.
patent: 4983596 (1991-01-01), Murata et al.
patent: 5093328 (1992-03-01), Sunagawa et al.
Chemical Abstracts vol. 18(23)233767(a) 1994.
Chemical Abstracts vol. 118:233767 (1983).
Chemical Abstracts vol. 118 233767(1993).

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Intermediaties for aminooxypyrrolidinylthiocarbapenem compounds does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Intermediaties for aminooxypyrrolidinylthiocarbapenem compounds, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Intermediaties for aminooxypyrrolidinylthiocarbapenem compounds will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-384388

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.