Intermediates useful in the preparation of diaminothiazoles

Details Intermediates useful in the preparation of diaminothiazoles Intermediates useful in the preparation of diaminothiazoles

2006-09-12

2006-09-12

Pryor, Alton (Department: 1616)

Organic compounds -- part of the class 532-570 series

Organic compounds

Nitrogen attached directly or indirectly to the purine ring...

C544S367000

Reexamination Certificate

active

07105670

ABSTRACT:
Disclosed are novel diaminothiazoles that are selective inhibitors of Cdk4. These compounds and their pharmaceutically acceptable salts and esters are anti-proliferative agents useful in the treatment or control of solid tumors, in particular breast, colon, lung and prostate tumors. Also disclosed are pharmaceutical compositions containing these compounds as well as intermediates useful in the preparation of the compounds.

REFERENCES:
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