Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1989-10-10
1992-05-05
Shah, Mukund J.
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
549331, 558429, 560117, C07D30794, C07D25704, C07C 69608
Patent
active
051109395
ABSTRACT:
Invented are 4-aza-5-alpha-8(14)-17 substituted-androsten-3-ones having an 8(14), 7(8), or 16(17) double bond, optionally also having a 1(2) double bond, pharmaceutical compositions containing the compounds, and methods of using these compounds to inhibit steroid 5-alpha-reductase.
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Holt Dennis A.
Levy Mark A.
Metcalf Brian W.
Dustman Wayne J.
Lentz Edward T.
Shah Mukund J.
SmithKline Beecham Corporation
Suter Stuart R.
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