Intermediates for preparing 1,6-dicarba-vasopressin compounds

Details Intermediates for preparing 1,6-dicarba-vasopressin compounds Intermediates for preparing 1,6-dicarba-vasopressin compounds

1988-05-09

1990-03-13

Shippen, Michael L.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carboxylic acid esters

560 12, 560 17, 560121, 560125, 562430, 562431, 562503, 562507, C07C125065

Patent

active

049084755

ABSTRACT:
New compounds which have potent V.sub.2 -vasopressin antagonistic activity are prepared by a 1,6-cyclization using peptide bond formation. The structures of the compounds are characterized by a Pas.sup.1,6 or Tas.sup.1,6 cyclized unit. Also a chiral synthesis of the optically pure Pas intermediates is described.

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