Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1993-05-13
1995-01-03
Ford, John M.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
544326, 544327, 544328, 544329, 544225, 544229, 544122, C07D23942, C07D40712, C07D40912, A01N 4354
Patent
active
053787080
DESCRIPTION:
BRIEF SUMMARY
BACKGROUND OF THE INVENTION
1. Field of the Invention
This invention concerns aralkylamino-pyrimidines, pesticidal compositions containing said compounds and use of the compounds to control pests.
2. State of the Art
U.S. Pat. No. 4,895,849 discloses aralkylaminopyrimidine derivatives of Formula I as insecticides, acaricides and fungicides ##STR2## wherein: A is an alkylene group optionally substituted with one or two substituents selected from the group alkynyl, haloalkyl, alkoxy, alkylthio and C.sub.3 -C.sub.5 cycloalkyl. ##STR3## wherein: R.sub.5 is H, lower alkyl, cycloalkyl or lower haloalkyl.
EP 323,757 discloses alkylaminopyrimidine derivatives, process for producing the same, and insecticide, acaricide and fungicides containing the same as an active ingredient.
U.S. Pat. No. 4,435,402 discloses aminopyrimidine derivatives, processes for their preparation, and fungicidal, insecticidal and acaricidal compositions containing them.
EP 196,524 discloses phenoxyalkylamino-pyrimidine derivatives.
SUMMARY OF THE INVENTION
The invention pertains to compounds of Formula I, including all geometric and stereoisomers, agriculturally suitable salts thereof, agricultural compositions containing them and their use as insecticides, acaricides and fungicides in both agronomic and nonagronomic environments. The compounds of the invention are: ##STR4## wherein: Q is selected from the group ##STR5## A is selected from the group C.sub.1 -C.sub.5 alkylene and C.sub.3 -C.sub.6 cycloalkylene, where any one atom of A can be optionally substituted with R.sup.1 ; C(O)R.sup.8, CO.sub.2 R.sup.8, C(O)N(R.sup.8)R.sup.9, N.sub.3, NO.sub.2, N(R.sup.8)R.sup.9, N(R.sup.8)C(O)R.sup.9, N(R.sup.8)C(O)N(R.sup.10)R.sup.9, N(R.sup.8)S(O).sub.2 R.sup.10, OR.sup.8. OC(O)R.sup.8, OCO.sub.2 R.sup.8, OC(O)N(R.sup.8)R.sup.9, OS(O).sub.2 R.sup.8, SR.sup.8, S(O)R.sup.8, S(O).sub.2 R.sup.8 and SCN; provided that when R.sup.1 is N(R.sup.8)S(O).sub.2 R.sup.10, then R.sup.10 is other than H and when R.sup.1 is OC(O)R.sup.8, OCO.sub.2 R.sup.8, OS(O).sub.2 R.sup.8, S(O)R.sup.8 or S(O).sub.2 R.sup.8, then R.sup.8 is other than H; C.sub.1 -C.sub.4 haloalkyl; C.sub.1 -C.sub.6 haloalkyl, C.sub.2 -C.sub.6 alkoxyalkyl and C.sub.2 -C.sub.6 alkylthioalkyl; -C.sub.6 haloalkyl, C.sub.2 -C.sub.6 alkoxyalkyl and C.sub.2 -C.sub.6 alkylthioalkyl; C.sub.2 -C.sub.6 alkylcarbonyl, C.sub.2 -C.sub.6 alkoxycarbonyl, C.sub.2 -C.sub.6 haloalkoxycarbonyl, C(O)R.sup.15, R.sup.11 OC(O)N(R.sup.12)S--, R.sup.11 (R.sup.12)NS--, and SR.sup.8 ; or R.sup.5 is C.sub.1 -C.sub.6 alkyl optionally substituted with a group selected from halogen, CN, NO.sub.2, S(O).sub.n R.sup.11, C(O)R.sup.11, CO.sub.2 R.sup.11, C.sub.1 -C.sub.3 haloalkoxy and phenyl optionally substituted by halogen, CN, or C.sub.1 -C.sub.2 haloalkyl; -C.sub.6 alkoxy, C.sub.2 -C.sub.6 alkoxyalkyl, C.sub.2 -C.sub.6 alkoxyalkoxy, C.sub.2 -C.sub.6 alkenyl, C.sub.2 -C.sub.6 haloalkenyl, C.sub.2 -C.sub.6 alkynyl, C.sub.2 -C.sub.6 alkenyloxy, C.sub.2 -C.sub.6 alkynyloxy, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 cycloalkylalkyl, C.sub.1 -C.sub.6 alkylthio, C.sub.1 -C.sub.6 alkylsulfinyl, C.sub.1 -C.sub.6 alkylsulfonyl, C.sub.1 -C.sub.6 haloalkylthio, C.sub.1 -C.sub.6 haloalkylsulfinyl, C.sub.1 -C.sub.6 haloalkylsulfonyl, phenyl optionally substituted with W and phenoxy optionally substituted with W; -C.sub.2 alkyl, C.sub.1 -C.sub.2 alkoxy and CF.sub.3 ; -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.2 -C.sub.6 haloalkenyl, C.sub.2 -C.sub.6 alkynyl, C.sub.3 -C.sub.6 haloalkynyl, C.sub.2 -C.sub.6 alkoxyalkyl, C.sub.2 -C.sub.6 alkylthioalkyl, C.sub.1 -C.sub.6 nitroalkyl, C.sub.2 -C.sub.6 cyanoalkyl, C.sub.3 -C.sub.8 alkoxycarbonylalkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 halocycloalkyl, phenyl optionally substituted with 1 to 3 substituents independently selected from W and benzyl optionally substituted with 1 to 3 substituents independently selected from W; --(CH.sub.2).sub.4 --, --(CH.sub.2).sub.5 -- or --CH.sub.2 CH.sub.2 OCH.sub.2 CH.sub.2 --; -C.sub.4 alkyl; -C.sub.4 alkoxyalkyl
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Kristiansen et al, Chemical Abstracts, vol. 117, entry 7945e (1992).
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Drumm, III Joseph E.
Lett Renee M.
Stevenson Thomas M.
Costello James A.
E. I. Du Pont de Nemours and Company
Ford John M.
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