Inhibitors of platelet-derived growth factor

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514246, 544180, 548427, 548451, 548475, 548477, A61K 3140, C07D20948

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active

052389502

ABSTRACT:
A method of inhibiting the binding of PDGF using compounds of the formula I ##STR1## useful in the treatment of atherosclerosis, cancer, retinal detachment, pulmonary fibrosis, arthritis, psoriasis and glomerulonephritis, and restenosis following angioplasty or vascular surgery is disclosed.
Also disclosed are pharmaceutical compositions and novel PDGF inhibitory compounds of the formula ##STR2## or a pharmaceutically acceptable addition salt thereof, useful in the treatment of atherosclerosis, cancer, retinal detachment, pulmonary fibrosis, arthritis, psoriasis and glomerulonephritis, and restenosis following angioplasty or vascular surgery.

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patent: 4194982 (1980-03-01), Chou
patent: 4266078 (1981-05-01), Pallos
Lukovits, Chemical Abstract, vol. 110(111, 1988, #87980f).
Soai, et al., Bull. Chem. Soc. Jpn., 55 1982) 1671-1672.
Ferns, et al., Science, 253 (1991) 1129-1132.

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