Inhibitors of cruzipain and other cysteine proteases

Details Inhibitors of cruzipain and other cysteine proteases Inhibitors of cruzipain and other cysteine proteases

2006-11-07

2006-11-07

Lambkin, Deborah C. (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C549S475000

Reexamination Certificate

active

07132449

ABSTRACT:
Compounds of general formula (I):wherein R1, R2, Y, (X)o, (W)n, (V)m, Z and U are as defined in the specification, are inhibitors of cruzipain and other cysteine protease inhibitors and are useful as therapeutic agents, for example in Chagas' disease, or for validating therapeutic target compounds.

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