Indolylalkylamino-methylidenecarbamate derivatives useful as...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C548S469000, C548S494000, C548S495000, C514S415000, C514S419000, C546S268100, C546S276400, C544S336000, C544S358000, C544S359000

Reexamination Certificate

active

07449489

ABSTRACT:
The invention relates to a group of novel indole compounds of Formula (I): wherein: R1, R2, R4, R6, R6a, R7, R8, R9, R10, and A are as defined in the specification, which are useful as gonadotrophin releasing hormone antagonists. The invention also relates to pharmaceutical formulations of said compounds, methods of treatment using said compounds and to processes for the preparation of said compounds.

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