Indole derivatives as H3 inverse agonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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Details

C514S414000, C514S217040, C514S228200, C514S235200, C514S316000, C514S323000, C540S597000, C544S124000, C544S144000, C546S187000, C546S201000, C548S468000

Reexamination Certificate

active

11157093

ABSTRACT:
The present invention relates to compounds of formula I:wherein X, R1, R2, R3, R4and R5are as defined in the description and claims, and pharmaceutically acceptable salts thereof, to the preparation of such compounds and pharmaceutical compositions containing them. The compounds are useful for the treatment and/or prevention of diseases which are associated with the modulation of H3 receptors.

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