Indole derivatives

Details Indole derivatives Indole derivatives

2007-07-26

2010-12-14

Jiang, Shaojia Anna (Department: 1623)

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

C514S043000

Reexamination Certificate

active

07851617

ABSTRACT:
Novel indole derivatives of formula (I) or a pharmaceutically acceptable salt thereof:wherein R1is fluorine, or chlorine, and R2is hydrogen, or fluorine, which are SGLT inhibitors and are useful for treatment or prevention of diabetes and related conditions.

REFERENCES:
patent: 5424406 (1995-06-01), Tsujihara et al.
patent: 5731292 (1998-03-01), Tsujihara et al.
patent: 5830873 (1998-11-01), Tsujihara et al.
patent: 6414126 (2002-07-01), Ellsworth et al.
patent: 6515117 (2003-02-01), Ellsworth et al.
patent: 6562791 (2003-05-01), Maurya et al.
patent: 2001/0041674 (2001-11-01), Tomiyama et al.
patent: 2002/0052326 (2002-05-01), Washburn
patent: 2002/0111315 (2002-08-01), Washburn et al.
patent: 2003/0064935 (2003-04-01), Gougoutas
patent: 2003/0087843 (2003-05-01), Washburn
patent: 2003/0114390 (2003-06-01), Washburn et al.
patent: 2004/0053855 (2004-03-01), Fujikura et al.
patent: 2004/0063646 (2004-04-01), Fujikura et al.
patent: 2004/0110936 (2004-06-01), Ohsumi et al.
patent: 2004/0116357 (2004-06-01), Fushimi et al.
patent: 2004/0132669 (2004-07-01), Nishimura et al.
patent: 2004/0138143 (2004-07-01), Glombik et al.
patent: 2004/0259819 (2004-12-01), Frick et al.
patent: 2005/0014704 (2005-01-01), Frick et al.
patent: 2005/0032711 (2005-02-01), Patel et al.
patent: 2005/0032712 (2005-02-01), Urbanski
patent: 2005/0037980 (2005-02-01), Rybczynski et al.
patent: 2005/0037981 (2005-02-01), Beavers et al.
patent: 2006/0217323 (2006-09-01), Patel et al.
patent: 2006/0229260 (2006-10-01), Rybczynski et al.
patent: 2006/0234954 (2006-10-01), Urbanski
patent: 2006/0293251 (2006-12-01), Urbanski et al.
patent: 2007/0060545 (2007-03-01), Nomura et al.
patent: 2008/0119422 (2008-05-01), Nomura et al.
patent: 2494177 (2004-02-01), None
patent: 203-06 (2006-05-01), None
patent: 1528066 (2005-05-01), None
patent: 1 803 729 (2007-07-01), None
patent: 2001-288178 (2001-10-01), None
patent: 2003-12686 (2003-01-01), None
patent: WO-01/27128 (2001-04-01), None
patent: WO-01/68660 (2001-09-01), None
patent: WO-01/74834 (2001-10-01), None
patent: WO-01/74835 (2001-10-01), None
patent: WO-02/053573 (2002-07-01), None
patent: WO-02/068439 (2002-09-01), None
patent: WO-02/068440 (2002-09-01), None
patent: WO-02/083066 (2002-10-01), None
patent: WO-02/088157 (2002-11-01), None
patent: WO-03/011880 (2003-02-01), None
patent: WO-03/020737 (2003-03-01), None
patent: WO-03/099836 (2003-12-01), None
patent: WO-2004/007517 (2004-01-01), None
patent: WO-2004/013118 (2004-02-01), None
patent: WO-2004/014931 (2004-02-01), None
patent: WO-2004/019958 (2004-03-01), None
patent: WO-2004/0052902 (2004-06-01), None
patent: WO-2004/052903 (2004-06-01), None
patent: WO-2004/080990 (2004-09-01), None
patent: WO-2005/012326 (2005-02-01), None
patent: WO-2006/035796 (2006-04-01), None
R.H.Unger et al., Diabetologia, vol. 28, (1985), pp. 119-121.
Luciano Rossetti M.D. et al.,Diabetes Care, vol. 13, No. 6, (Jun. 1990), pp. 610-630.
Luciano Rossetti et al.,J. Clin. Invest., vol. 79, (May 1987), pp. 1510-1515.
Luciano Rossetti et al.,J. Clin. Invest.., vol. 80, (Oct. 1987), pp. 1037-1044.
Barbara B. Kahn et al.,J. Clin Invest., vol. 87, (Feb. 1991), pp. 561-570.
Kenji Tsujihara et al.,J. Med. Chem., vol. 42, (1999), pp. 5311-5324.
Kenji Arakawa et al.,British Journal of Pharmacology, vol. 132, (2001), pp. 578-586.
Ahmad et al.,Nucleosides, Nucleotides&Nucleic Acids, vol. 20, No. 9, (2001), pp. 1671-1682.
Zamani et al.,Journal of the Chinese Chemical Society, vol. 49, (2002), pp. 1041-1044.
Maatooq et al.,Phytochemistry, vol. 44, No. 1, (Jan. 1997), pp. 187-190.
Hongu et al., Chem. Pharm. Bull., vol. 46, No. 1, pp. 22-33, (1998).

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