Indazole derivatives as CRF antagonists

Details Indazole derivatives as CRF antagonists Indazole derivatives as CRF antagonists

2007-05-08

2007-05-08

Stockton, Laura L. (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S405000, C548S362100, C548S361100, C548S362500

Reexamination Certificate

active

10724971

ABSTRACT:
This invention relates to compounds which are generally CRF-1 receptor antagonists and which are represented by Formula I or Formula II:wherein R3is optionally substituted aryl or heteroaryl, R1and R2are as defined in the specification; or individual isomers, racemic or non-racemic mixtures of isomers, or pharmaceutically acceptable salts thereof. The invention further relates to processes for preparing such compounds, to pharmaceutical compositions containing such compounds, and to methods for their use as therapeutic agents.

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