Immunosuppressive fluorinated cyclosporin analogs

Details Immunosuppressive fluorinated cyclosporin analogs Immunosuppressive fluorinated cyclosporin analogs

1991-04-29

1993-07-13

Chan, Y. Christina

Chemistry: natural resins or derivatives; peptides or proteins;

Peptides of 3 to 100 amino acid residues

Cyclic peptides

530317, C07K 764, A61K 3702

Patent

active

052274675

ABSTRACT:
New immunosuppressive cyclosporin analogs are disclosed having one or more fluorinated amino acids. These analogs may also have a "C-9 amino acid" wherein the double bond is replaced by a heteroatom such as sulfur or oxygen.

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