Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1993-11-15
1995-02-07
Shah, Mukund J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
540555, 540558, 540560, 540562, A61K 3155, C07D48714, C07D49522
Patent
active
053875850
ABSTRACT:
The novel imidazodiazepine derivatives of the formula: ##STR1## wherein the substituents are as described in the specification, can be used for the control or prevention of epileptic seizures, anxiety, tension and excitation states, sleep disorders, schizophrenic symptoms, hepatic encephalopathy and senile dementia, as well as, in the partial or complete antagonization of undesired side-effects of substances acting on benzodiazepine receptors after over-dosage or after their use in intensive medicine and in anesthesia.
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Borer Rene
Gassner Walter
Gerecke Max
Kyburz Emilio
Ciambrone Coletti Ellen
Datlow Philip I.
Gould George M.
Hoffmann-La Roche Inc.
Johnston George W.
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