Hydrolytic enzyme inhibitors/inactivators and methods for using

Details Hydrolytic enzyme inhibitors/inactivators and methods for using Hydrolytic enzyme inhibitors/inactivators and methods for using

1995-02-14

1996-10-22

Kight, John

Chemistry: molecular biology and microbiology

Measuring or testing process involving enzymes or...

Involving hydrolase

435 4, 435 19, 435188, 435195, 435198, 435232, 435184, 554 78, 554 79, 554 80, 534727, 534852, 558179, C12Q 134, C12Q 100, C12N 996, C07F 902

Patent

active

055675972

ABSTRACT:
The present invention provides compounds that function as hydrolytic enzyme inhibitors (inactivators) and substrates. These compounds are useful in assays to detect and measure levels of hydrolytic enzyme activity and are more particularly useful in treatment regimens for various disease states and conditions implicating the underlying specific hydrolytic enzyme. Examples of hydrolytic enzymes include, but are not limited to, phospholipases, lipases, esterases, proteases, etc.

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