Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1994-08-23
1996-03-26
McKane, Joseph K.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
5142334, 514432, 514621, 544162, 544145, 549 23, 564169, 564164, 564163, 564158, 564155, A61K 31395, C07D26528
Patent
active
055020534
ABSTRACT:
Compounds of formula ##STR1## are HIV protease inhibitors, and are synthesized via a novel route. These compounds are useful in the prevention or treatment of infection by HIV and in the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ingredients, whether or not in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of treating AIDS and methods of preventing or treating infection by HIV are also described.
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Britcher Susan F.
Dorsey Bruce D.
Huff Joel R.
McKane Joseph K.
Merck & Co. , Inc.
Meredith Roy D.
Quagliato Carol S.
Winokur Melvin
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