Histamine H.sub.3 -receptor antagonists and therapeutic uses the

Details Histamine H.sub.3 -receptor antagonists and therapeutic uses the Histamine H.sub.3 -receptor antagonists and therapeutic uses the

1994-06-15

1997-05-27

Reamer, James H.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

5483147, 546203, C07D41100

Patent

active

056333820

ABSTRACT:
The present invention provides novel compounds having activity as histamine H.sub.3 -receptor antagonists. The novel compounds include 4-imidazolyl-N-substituted pyrrolidines, piperidines, and cycloheptimides. The preferred compounds are 4-imidazolyl-N-(cycloalkyl/aryl-alkyl-carbonyl) piperidines such as 4-(1-cyclohexylvaleryol-4-piperidyl)-1H-imidazole.

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